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valerenic acid/psychomotor agitation

Veza se sprema u međuspremnik
ČlanciKliničkim ispitivanjimaPatenti
2 rezultati
Valerian extracts have been used for centuries to alleviate restlessness and anxiety albeit with unknown mechanism of action in vivo. We now describe a specific binding site on GABA(A) receptors with nM affinity for valerenic acid and valerenol, common constituents of valerian. Both agents enhanced

Valerian extract and valerenic acid are partial agonists of the 5-HT5a receptor in vitro.

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Insomnia is the most frequently encountered sleep complaint worldwide. While many prescription drugs are used to treat insomnia, extracts of valerian (Valeriana officinalis L., Valerianaceae) are also used for the treatment of insomnia and restlessness. To determine novel mechanisms of action,
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