Anti-cancer drug design
New cytotoxic analogues of annonaceous acetogenins.
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Přihlášení Registrace
Odkaz je uložen do schránky
Klíčová slova
Abstraktní
A series of new acetogenin analogues incorporating a central catechol moiety instead of the tetrahydrofuran ring(s) have been prepared and tested against L1210 leukemia cells. Although less potent than bullatacinone, which has the same terminal lactone, these compounds display interesting cell cycle effects.