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ascaridole/malaria

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Mechanism of ascaridole activation in Leishmania.

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Endoperoxides (EP) are an emerging class of drugs which have potential in antiparasitic therapy, but also in other fields. For malaria therapy the EP artemisinin (Art) and its derivatives are successfully used. We have shown in the past that the EP ascaridole (Asc) is useful for the treatment of

Activation of Artemisinin and Heme Degradation in Leishmania tarentolae Promastigotes: A Possible Link.

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Endoperoxides (EPs) appear to be promising drug candidates against protozoal diseases, including malaria and leishmaniasis. Previous studies have shown that these drugs need an intracellular activation to exert their pharmacological potential. The efficiency of these drugs is linked to the extensive

Chemical composition and insecticidal activity of plant essential oils from Benin against Anopheles gambiae (Giles).

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BACKGROUND Insecticide resistance in sub-Saharan Africa and especially in Benin is a major public health issue hindering the control of the malaria vectors. Each Anopheles species has developed a resistance to one or several classes of the insecticides currently in use in the field. Therefore, it is
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