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soyasapogenol b/lifrarbólga

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GreinarKlínískar rannsóknirEinkaleyfi
3 niðurstöður

Preventive effects of soyasapogenol B derivatives on liver injury in a concanavalin A-induced hepatitis model.

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To shed light on the structure-activity relationship, various soyasapogenol B derivatives were synthesized and evaluated for preventive effects on liver injury in the concanavalin A (Con A)-induced hepatitis model in mice. Con A injection into mice induces some pathophysiology of human liver disease
OBJECTIVE ME3738, a derivative of soyasapogenol B, enhances the anti-hepatitis C virus (HCV) effect of interferon in an in vitro replication system and an in vivo mouse model of HCV infection. ME3738 plus pegylated interferon (PEG IFN)-α-2a treatment for 12 weeks decreased HCV RNA levels in enrolled

ME3738 enhances the effect of interferon and inhibits hepatitis C virus replication both in vitro and in vivo.

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OBJECTIVE ME3738 (22β-methoxyolean-12-ene-3β, 24-diol), a derivative of soyasapogenol B, attenuates liver disease in several animal models of acute and chronic liver injury. ME3738 is thought to inhibit replication of hepatitis C virus (HCV) by enhancing interferon (IFN)-β production, as determined
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