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bruceantin/pykinimas

Nuoroda įrašoma į mainų sritį
StraipsniaiKlinikiniai tyrimaiPatentai
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Initial clinical studies with bruceantin.

Straipsnius versti gali tik registruoti vartotojai
Prisijungti Registracija
A phase I clinical study of bruceantin was conducted in 66 patients with various types of advanced solid tumors to evaluate its toxicity and efficacy. The initial dose of 0.2 mg/m2/day x 5 days repeated at 2-week intervals was progressively increased to a maximum dose of 4.5 mg/m2/day. Hypotension

Phase I study on bruceantin administered on a weekly schedule.

Straipsnius versti gali tik registruoti vartotojai
Prisijungti Registracija
Fifteen adult patients with advanced solid tumors received bruceantin at doses of 1.6-6.0 mg/m2 iv for 30 minutes/week X 4, followed by a 2-week rest. The dose-limiting toxic effect was nausea and vomiting, which was more severe in patients with hepatic metastases or liver function abnormalities.

Clinical pharmacology of bruceantin by radioimmunoassay.

Straipsnius versti gali tik registruoti vartotojai
Prisijungti Registracija
During the phase I clinical trial of a new antitumor agent, bruceantin, the pharmacology was studied in 18 cancer patients. The drug was infused intravenously (IV) for 3 h at doses ranging from 1 to 3.6 mg/m2 per day for 5 days. The plasma drug disappearance curves were biphasic, with a fast initial

A Phase II study of Bruceantin (NSC-165, 563) in advanced malignant melanoma.

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Prisijungti Registracija
The Eastern Cooperative Oncology Group (ECOG) conducted a Phase II trial of Bruceantin in malignant melanoma. Twenty-two patients, thirteen without prior cytotoxic chemotherapy, were entered. All patients were evaluable for response and toxicity. Dose limiting toxicity was found to be hypotension

Phase II trial of bruceantin in metastatic breast carcinoma.

Straipsnius versti gali tik registruoti vartotojai
Prisijungti Registracija
A phase II evaluation of bruceantin was carried out in 15 patients with refractory metastatic breast cancer. All patients had received extensive prior therapy including adriamycin, cytoxan, 5-FU, methotrexate, and a vinca alkaloid. Except for two patients with stable disease, no complete or partial
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