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phyllanthoside/rhabdomyosarcoma

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ČlankiKliničnih preskušanjPatenti
2 rezultatov

Isolation, identification and biological activity of a phyllanthoside metabolite produced in vitro by mouse plasma.

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Prijava / prijava
The antitumor agent phyllanthoside is rapidly metabolized in vitro by mouse plasma. This metabolite has now been isolated from mouse plasma and its structural properties and cytotoxicity characterized. The isolated metabolite was estimated to be greater than 98% pure by HPLC analysis. Mass spectral

Disposition and metabolism of the antitumor glycoside phyllanthoside in mouse and beagle dog.

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Prijava / prijava
Phyllanthoside is a naturally occurring glycoside with activity against IP transplantable murine tumors. Phyllanthoside administered IV, to mice at a nontoxic dose of 16 mg/kg could not be detected in blood or plasma even 30 s after administration. There was rapid formation of a less polar
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