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Natural Product Research 2006-Apr

Biflavonoids inhibited phosphatase of regenerating liver-3 (PRL-3).

Watumiaji waliosajiliwa tu ndio wanaweza kutafsiri nakala
Ingia / Ingia
Kiungo kimehifadhiwa kwenye clipboard
Sung-Kyu Choi
Hyun-Mi Oh
Su-Kyung Lee
Dae Gwin Jeong
Seong Eon Ryu
Kwang-Hee Son
Dong Cho Han
Nack-Do Sung
Nam-In Baek
Byoung-Mog Kwon

Maneno muhimu

Kikemikali

Two biflavonoids, ginkgetin (1) and sciadopitysin (2), were isolated from the MeOH extract of the young branches of Taxus cuspidata, which inhibited phosphatase of regenerating liver-3 (PRL-3) with IC50 values of 25.8 and 46.2 microM, respectively. This is the first report on PRL-3 inhibitors, isolated from natural sources.

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