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diterpene lactone/breast neoplasms

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NakalaMajaribio ya klinikiHati miliki
3 matokeo
Matrix metalloproteinase-9 (MMP-9) plays a critical role in cancer metastasis. Andrographolide (AP) is a diterpene lactone in the leaves and stem of Andrographis paniculata (Burm. f) Ness that has been reported to possess anticancer activity. In this study, we investigated the effect of AP on

mPEG-PLA Micelle for Delivery of Effective Parts of Andrographis Paniculata.

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Ingia / Ingia
BACKGROUND Many studies have shown that Andrographis paniculata (Burm. f.) Nees has a good anti-tumor effect, but poor solubility in water and poor bioavailability hinder the modernization of it. METHODS To formulate the effective parts (mainly diterpene lactones) of Andrographis paniculata (AEP)

Anticancer activity of andrographolide semisynthetic derivatives.

Watumiaji waliosajiliwa tu ndio wanaweza kutafsiri nakala
Ingia / Ingia
Andrographolide 1, a diterpene lactone of Andrographis paniculata, displays in vitro and in vivo antitumor activity against breast cancer models and mouse myeloid leukemia (M1) cells. In the present study, we report the semi-synthesis of andrographolide derivatives and their in vitro activity
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